Abstract
Selenium is an essential micronutrient that is beneficial to human health. Selenium-containing drugs have been developed as antioxidants, anti-inflammatory, and anticancer agents. However, the synthesis of selenium-containing chalcones has not been fully explored. Therefore, we report the synthesis of novel selenophene-based chalcone analogs and reveal their biological activities as anticancer agents. Among the seven synthesized molecules, compounds 6, 8, and 10 exhibited anticancer activity with IC50 values of 19.98 ± 3.38, 38.23 ± 3.30, and 46.95 ± 5.68 μM, respectively, against human colorectal adenocarcinoma (HT-29) cells. Clonogenic assays and Western blot analysis tests further confirmed that compound 6 effectively induced apoptosis in HT-29 cells through mitochondrial- and caspase-3-dependent pathways.
Original language | English |
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Article number | 2200486 |
Pages (from-to) | e2200486 |
Journal | Archiv der Pharmazie |
Volume | 356 |
Issue number | 4 |
DOIs | |
State | Published - 04 2023 |
Externally published | Yes |
Bibliographical note
© 2022 Deutsche Pharmazeutische Gesellschaft.Keywords
- anticancer
- chalcone
- human colorectal adenocarcinoma cell
- selenophene
- Cell Proliferation
- Humans
- Structure-Activity Relationship
- Chalcones/pharmacology
- Chalcone
- Selenium/pharmacology
- Antineoplastic Agents/pharmacology
- Cell Line, Tumor
- Molecular Structure
- Apoptosis
- Drug Screening Assays, Antitumor