Leveraging a Low-Affinity Diazaspiro Orthosteric Fragment to Reduce Dopamine D3 Receptor (D3R) Ligand Promiscuity across Highly Conserved Aminergic G-Protein-Coupled Receptors (GPCRs)

  • Sean W. Reilly
  • , Aladdin A. Riad
  • , Chia Ju Hsieh
  • , Kristoffer Sahlholm
  • , Daniel A. Jacome
  • , Suzy Griffin
  • , Michelle Taylor
  • , Chi Chang Weng
  • , Kuiying Xu
  • , Nathan Kirschner
  • , Robert R. Luedtke
  • , Christopher Parry
  • , Shipra Malhotra
  • , John Karanicolas
  • , Robert H. Mach*
  • *此作品的通信作者

研究成果: 期刊稿件文章同行評審

19 引文 斯高帕斯(Scopus)

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Pharmacology, Toxicology and Pharmaceutical Science

Biochemistry, Genetics and Molecular Biology